Krogsgaard-Larsen, Povl.

Textbook of drug design and discovery / edited by Povl Krogsgaard-Larsen, Kristian Strømgaard, Ulf Madsen. - 4th ed. - Boca Raton, FL : CRC Press/Taylor & Francis, c2010. - xv, 460 p. : ill. (some col.) ; 27 cm.

Includes bibliographical references and index.

Molecular recognition in ligand-protein binding / Tommy Liljefors -- Biostructure-based drug design / Flemming S. Jørgensen and Jette S. Kastrup -- Ligand-based drug design / Ingrid Pettersson, Thomas Balle, and Tommy Liljefors -- Chemical biology / Kristian Strømgaard -- Stereochemistry in drug design / M. Belen Mayo-Martin and David E. Jane -- Natural products in drug discovery / Guy T. Carter -- Imaging in drug discovery and development / Markus Rudin and Thomas Mueggler -- Peptides and peptidomimetics / Minying Cai, Vinod Kulkarni, and Victor J. Hruby -- Prodrugs : design and development / Anders Buur and Niels Mørk -- Metals in medicine : inorganic medicinal chemistry / Helle R. Hansen and Ole Farver -- Enzyme inhibitors : biostructure-based and mechanism-based designs / Robert A. Copeland, Richard R. Gontarek, and Lusong Luo -- Receptors : structure, function, and pharmacology / Hans Bräuner-Osborne -- Ion channels : structure and function / Søren-Peter Olesen and Daniel B. Timmermann -- Neurotransmitter transporters : structure and function / Claus J. Loland and Ulrik Gether -- GABA and glutamic acid receptor ligands / Bente Frølund and Ulf Madsen -- Acetylcholine / Anders A. Jensen and Povl Krogsgaard-Larsen -- Histamine receptors / Iwan de Esch, Henk Timmerman and Rob Leurs -- Dopamine and serotonin / Benny Bang-Andersen and Klaus P. Bøgesø -- Opioid and cannabinoid receptors / Rasmus P. Clausen and Harald S. Hansen -- Hypnotics / Bjarke Ebert and Keith Wafford -- Neglected diseases / Søren B. Christensen -- Immunomodulating agents / Ulla G. Sidelmann -- Anticancer agents / Fredrik Bjørkling and Lars H. Jensen -- Antiviral drugs / Erik De Clercq -- Antibiotics / Piet Herdewijn.

9781420063226 (alk. paper) 1420063227 (alk. paper) 9781420063264 (alk. paper) 142006326X (alk. paper)

2009013698

GBA965109 bnb

101500606 DNLM 015302612 Uk


Drugs--Design.
Drug Design.
Drug Discovery.

RS420 / .T49 2010

615.1